PDBID: 3QTFTitle: DESIGN AND SAR OF MACROCYCLIC HSP90 INHIBITORS WITH INCREASED
METABOLIC STABILITY AND POTENT CELL-PROLIFERATION ACTIVITY
Molecule: HEAT SHOCK PROTEIN HSP 90-ALPHA Chain: A Fragment: N-TERMINAL DOMAIN (UNP RESIDUES 10-236) Organism: HOMO SAPIENS Method: X-RAY DIFFRACTION First author: C.W.ZAPF Resolution[Å]: 1.57 R-VALUE: 0.187 |
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