PDBID: 3R92Title: DISCOVERY OF A MACROCYCLIC O-AMINOBENZAMIDE HSP90 INHIBITOR WITH
HETEROCYCLIC TETHER THAT SHOWS EXTENDED BIOMARKER ACTIVITY AND IN
VIVO EFFICACY IN A MOUSE XENOGRAFT MODEL.
Molecule: HEAT SHOCK PROTEIN HSP 90-ALPHA Chain: A Fragment: N-TERMINAL DOMAIN, UNP RESIDUES 10-236 Organism: HOMO SAPIENS Method: X-RAY DIFFRACTION First author: C.W.ZAPF Resolution[Å]: 1.58 R-VALUE: 0.176 |
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