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Sep. 10, 2014:
A total of 174 experimentally verified S-nitrosylation sites on 94 S-nitrosylated proteins from individualized human colorectal cancer tissues using a label-free quantitation strategy.

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PDBID: 3R92

Title: DISCOVERY OF A MACROCYCLIC O-AMINOBENZAMIDE HSP90 INHIBITOR WITH HETEROCYCLIC TETHER THAT SHOWS EXTENDED BIOMARKER ACTIVITY AND IN VIVO EFFICACY IN A MOUSE XENOGRAFT MODEL.

Molecule: HEAT SHOCK PROTEIN HSP 90-ALPHA

Chain: A

Fragment: N-TERMINAL DOMAIN, UNP RESIDUES 10-236

Organism: HOMO SAPIENS

Method: X-RAY DIFFRACTION

First author: C.W.ZAPF

Resolution[Å]: 1.58

R-VALUE: 0.176

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